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Target
Vitamin K epoxide reductase complex subunit 1
Ligand
BDBM50015558
Substrate
n/a
Meas. Tech.
ChEBML_214470
Ki
100000±n/a nM
Citation
 Ryall, RP; Nandi, DL; Silverman, RB Substituted vitamin K epoxide analogues. New competitive inhibitors and substrates of vitamin K1 epoxide reductase. J Med Chem 33:1790-7 (1990) [PubMed]
Target
Name:
Vitamin K epoxide reductase complex subunit 1
Synonyms:
VKOR1_BOVIN | VKORC1 | Vitamin k epoxide reductase complex subunit 1 isoform 1
Type:
PROTEIN
Mol. Mass.:
17977.60
Organism:
Bos taurus
Description:
ChEMBL_305987
Residue:
163
Sequence:
MGATWRSPGWVRLALCLAGLVLSLYALHVKAARARDRDYRALCDVGTAISCSRVFSSRWGRGFGLVEHVLGKDSILNQSNSIFGCIFYTLQLLLGCLQGRWASVLLRLSCLVSLAGSVYLAWILFFVLYDFCIVCITTYAINVGLTVLSFREVQGPQGKVKGH
  
Inhibitor
Name:
BDBM50015558
Synonyms:
1a-(1-Fluoro-3,7,11,15-tetramethyl-hexadecyl)-7a-methyl-1a,7a-dihydro-1-oxa-cyclopropa[b]naphthalene-2,7-dione | CHEMBL50340
Type:
Small organic molecule
Emp. Form.:
C31H47FO3
Mol. Mass.:
486.7015
SMILES:
CC(C)CCCC(C)CCCC(C)CCCC(C)CC(F)C12OC1(C)C(=O)c1ccccc1C2=O
Structure:
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