Reaction Details
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Target
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial
Ligand
BDBM50486215
Substrate
n/a
Meas. Tech.
ChEMBL_894640 (CHEMBL3049710)
IC50
95380±n/a nM
Citation
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More Info.:
Target
Name:
Pyruvate dehydrogenase E1 component subunit alpha,/beta, mitochondrial
Synonyms:
Pyruvate dehydrogenase complex
Type:
n/a
Mol. Mass.:
n/a
Description:
ASSAY_ID of ChEMBL is 894639
Components:
This complex has 2 components.
Component 1
Name:
Pyruvate dehydrogenase E1 component subunit alpha, mitochondrial
Synonyms:
1.2.4.1 | ODPA_PEA | PDHE1-A | Pyruvate dehydrogenase E1 component subunit alpha, mitochondrial
Type:
PROTEIN
Mol. Mass.:
43536.99
Organism:
Pisum sativum
Description:
ChEMBL_106715
Residue:
397
Sequence:
MALSRLSSSSSSSNGSNLFNPFSAAFTLNRPISSDTTATLTIETSLPFTAHNCDPPSRSVTTSPSELLSFFRTMALMRRMEIAADSLYKANLIRGFCHLYDGQEAVAVGMEAGTTKKDCIITAYRDHCTFLGRGGTLLRVYAELMGRRDGCSKGKGGSMHFYKKDSGFYGGHGIVGAQVPLGCGLAFGQKYLKDESVTFALYGDGAANQGQLFEALNISALWDLPAILVCENNHYGMGTATWRSAKSPAYFKRGDYVPGLKVDGMDALAVKQACKFAKEHALKNGPIILEMDTYRYHGHSMSDPGSTYRTRDEISGVRQERDPIERVRKLLLSHDIATEKELKDTEKEVRKEVDEAIAKAKDSPMPDPSDLFSNVYVKGYGVEAFGVDRKEVRVTLP
Component 2
Name:
Pyruvate dehydrogenase E1 component subunit beta, mitochondrial
Synonyms:
1.2.4.1 | ODPB_PEA | PDHE1-B | Pyruvate dehydrogenase E1 component subunit beta, mitochondrial
Type:
PROTEIN
Mol. Mass.:
38791.52
Organism:
Pisum sativum
Description:
ChEMBL_106715
Residue:
359
Sequence:
MLGVIRNKTIRPSFSAFRFFSSAKQMTVRDALNSALDVEMSADSKVFLMGEEVGEYQGAYKVTKGLLEKYGPERVLDTPITEAGFTGIGVGAAYYGLKPVVEFMTFNFSMQAIDHIINSAAKSNYMSAGQISVPIVFRGLNGDAAGVGAQHSHCYASWYGSCPGLKVLVPHSAEDARGLLKAAIRDPDPVVFLENELLYGESFPVSAEVLDSSFWLPIGKAKIEREGKDVTITAFSKMVGFALKAAEILEKEGISAEVINLRSIRPLDRPTINASVRKTNRLVTVEEGFPQHGVGAEICTSVIEESFGYLDATVERIGGADVPMPYAGNLERLVVPHVEDIVRAAKRACHRSVPLAAAA