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Target
Probable G-protein coupled receptor 174
Ligand
BDBM50601676
Substrate
n/a
Meas. Tech.
ChEMBL_2237847 (CHEMBL5151743)
IC50
270±n/a nM
Citation
 Sayama, M; Uwamizu, A; Ikubo, M; Chen, L; Yan, G; Otani, Y; Inoue, A; Aoki, J; Ohwada, T Switching Lysophosphatidylserine G Protein-Coupled Receptor Agonists to Antagonists by Acylation of the Hydrophilic Serine Amine. J Med Chem 64:10059-10101 (2021) [PubMed]  Article
Target
Name:
Probable G-protein coupled receptor 174
Synonyms:
GP174_MOUSE | Gm376 | Gpr174
Type:
PROTEIN
Mol. Mass.:
38774.65
Organism:
Mus musculus
Description:
ChEMBL_116800
Residue:
335
Sequence:
MTDNFTCNKTDGDNTDFRYFIYAVTYTVILVPGLIGNILALWVFYGYMKETKRAVVFMINLAIADLLQILSLPLRIFYYLNHDWPFGPGLCMFCFYLKYVNMYASIYFLVCISVRRFWFLMYPFRFNDCKQKYDLYISIIGWLIICLACLLFPLLRTNDDTPGNRTKCFVDLPIRNVNLAQSVAMITIGEVVGFVTPLMIVLYCTWKTALSLQNKYPISQHLGEKKKALKMILTCAGVFLVCFVPYHFSFPLDFLVKSNEIKSCFARRVILIFHSVALCLASLNSCLDPVIYYFTTNEFRRRLSRQDLPDNIQLHTKSYKIASNHATSTVAAELC
  
Inhibitor
Name:
BDBM50601676
Synonyms:
CHEMBL5192494
Type:
Small organic molecule
Emp. Form.:
C28H47N2O9P
Mol. Mass.:
586.6545
SMILES:
CCCCCCCCCCCOc1cccc(CCC(=O)NCCCOP(O)(=O)OC[C@H](NC(C)=O)C(O)=O)c1 |r|
Structure:
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