Reaction Details
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Target
Trypanothione reductase
Ligand
BDBM50612874
Substrate
n/a
Meas. Tech.
ChEMBL_2290321
IC50
3600±n/a nM
Citation
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More Info.:
Target
Name:
Trypanothione reductase
Synonyms:
1.8.1.12 | N(1),N(8)-bis(glutathionyl)spermidine reductase | TPR | Trypanothione reductase
Type:
PROTEIN
Mol. Mass.:
53444.86
Organism:
Trypanosoma congolense
Description:
ChEMBL_120929
Residue:
492
Sequence:
MSKAFDLVIIGAGSGGLEAGWNAATLYKKRVAVVDVQTVHGPPFFAALGGTCVNVGCVPKKLMVTGAQYMDQLRESAGFGWEFDASTIKANWKTLIAAKNAAVLDINKSYEDMFKDTEGLEFFLGWGALEQKNVVTVREGADPKSKVKERLQAEHIIIATGSWPQMLKIPGIEHCISSNEAFYLEEPPRRVLTVGGGFISVEFAGIFNAYKPVGGKVTLCYRNNPILRGFDYTLRQELTKQLVANGIDIMTNENPSKIELNPDGSKHVTFESGKTLDVDVVMMAIGRLPRTGYLQLQTVGVNLTDKGAIQVDEFSRTNVPNIYAIGDVTGRIMLTPVAINEGASVVDTIFGSKPRKTDHTRVASAVFSIPPIGTCGLTEEEAAKSFEKVAVYLSCFTPLMHNISGSKYKKFVAKIITDHGDGTVVGVHLLGDSSPEIIQAVGICMKLNAKISDFYNTIGVHPTSAEELCSMRTPSHYYIKGEKMETLPDSSL