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Target
Fatty acid-binding protein 5
Ligand
BDBM212456
Substrate
n/a
Meas. Tech.
ChEMBL_2301983
IC50
3790±n/a nM
Citation
 Floresta, G; Pistarà, V; Amata, E; Dichiara, M; Marrazzo, A; Prezzavento, O; Rescifina, A Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review. Eur J Med Chem 138:854-873 (2017) [PubMed]
Target
Name:
Fatty acid-binding protein 5
Synonyms:
FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5)
Type:
Enzyme
Mol. Mass.:
15164.79
Organism:
Homo sapiens (Human)
Description:
Q01469
Residue:
135
Sequence:
MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTLKTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVECVMNNVTCTRIYEKVE
  
Inhibitor
Name:
BDBM212456
Synonyms:
US9278918, 46
Type:
Small organic molecule
Emp. Form.:
C19H18Cl2N2O3
Mol. Mass.:
393.264
SMILES:
OC(=O)C1(CCCC1)NC(=O)Nc1cc(Cl)cc(Cl)c1-c1ccccc1
Structure:
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