Reaction Details Report a problem with these data
Target
GTP:AMP phosphotransferase AK3, mitochondrial
Ligand
BDBM50367099
Substrate
n/a
Meas. Tech.
ChEMBL_32211 (CHEMBL875019)
Ki
3000000±n/a nM
Citation
Hai, TT; Picker, D; Abo, M; Hampton, A Species- or isozyme-specific enzyme inhibitors. 7. Selective effects in inhibitions of rat adenylate kinase isozymes by adenosine 5'-phosphate derivatives. J Med Chem 25:806-12 (1982) [PubMed]
More Info.:
Target
Name:
GTP:AMP phosphotransferase AK3, mitochondrial
Synonyms:
AK 3 | Adenylate kinase 3 | Adenylate kinase 3 alpha like 1 | Adenylate kinase 3 alpha-like 1 | Ak3 | Ak3l1 | Akl3l | GTP:AMP phosphotransferase mitochondrial | KAD3_RAT
Type:
PROTEIN
Mol. Mass.:
25443.58
Organism:
Rattus norvegicus
Description:
ChEMBL_1340551
Residue:
227
Sequence:
MGASGRLLRAVIMGAPGSGKGTGSSRITKHFELKHLSSGDLLRQNMLQGTEIAVLAKSFIDQGKLIPDDDMTRLALHELKNLTQCSWLLDGFPRTLPQAEALDRVYQIDTVINLNVPFEVIKLRLTARWIHPASGRVYNIEFNPPKTVGIDDLTGEPLIQREDDKPETVIKRLKAYEAQTEPVLQYYQKKGVLETFSGTETNKIRPHVYSFLQMKVPETIQKASVTP