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Target
Serine/threonine-protein kinase 32B
Ligand
BDBM50393108
Substrate
n/a
Meas. Tech.
ChEMBL_853871 (CHEMBL2154991)
Kd
40000±n/a nM
Citation
 Shengule, SR; Loa-Kum-Cheung, WL; Parish, CR; Blairvacq, M; Meijer, L; Nakao, Y; Karuso, P A one-pot synthesis and biological activity of ageladine A and analogues. J Med Chem 54:2492-503 (2011) [PubMed]  Article
Target
Name:
Serine/threonine-protein kinase 32B
Synonyms:
ST32B_HUMAN | STK32B | YANK2
Type:
PROTEIN
Mol. Mass.:
47892.49
Organism:
Homo sapiens (Human)
Description:
ChEMBL_587221
Residue:
414
Sequence:
MGGNHSHKPPVFDENEEVNFDHFQILRAIGKGSFGKVCIVQKRDTKKMYAMKYMNKQKCIERDEVRNVFRELQIMQGLEHPFLVNLWYSFQDEEDMFMVVDLLLGGDLRYHLQQNVHFTEGTVKLYICELALALEYLQRYHIIHRDIKPDNILLDEHGHVHITDFNIATVVKGAERASSMAGTKPYMAPEVFQVYMDRGPGYSYPVDWWSLGITAYELLRGWRPYEIHSVTPIDEILNMFKVERVHYSSTWCKGMVALLRKLLTKDPESRVSSLHDIQSVPYLADMNWDAVFKKALMPGFVPNKGRLNCDPTFELEEMILESKPLHKKKKRLAKNRSRDGTKDSCPLNGHLQHCLETVREEFIIFNREKLRRQQGQGSQLLDTDSRGGGQAQSKLQDGCNNNLLTHTCTRGCSS
  
Inhibitor
Name:
BDBM50393108
Synonyms:
CHEMBL2153266
Type:
Small organic molecule
Emp. Form.:
C15H11N5
Mol. Mass.:
261.2813
SMILES:
Nc1nc2c(nccc2[nH]1)-c1cnc2ccccc2c1
Structure:
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