Reaction Details Report a problem with these data
Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50035218
Substrate
n/a
Meas. Tech.
ChEMBL_1452788 (CHEMBL3365130)
IC50
810±n/a nM
Citation
Kamal, A; Srinivasa Reddy, T; Polepalli, S; Paidakula, S; Srinivasulu, V; Ganga Reddy, V; Jain, N; Shankaraiah, N Synthesis and biological evaluation of 4-aza-2,3-dihydropyridophenanthrolines as tubulin polymerization inhibitors. Bioorg Med Chem Lett 24:3356-60 (2014) [PubMed] Article
More Info.:
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP