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Target
Thiol:disulfide interchange protein DsbA
Ligand
BDBM50062489
Substrate
n/a
Meas. Tech.
ChEMBL_1462817 (CHEMBL3399656)
Kd
13100±n/a nM
Citation
Duprez, W; Premkumar, L; Halili, MA; Lindahl, F; Reid, RC; Fairlie, DP; Martin, JL Peptide inhibitors of the Escherichia coli DsbA oxidative machinery essential for bacterial virulence. J Med Chem 58:577-87 (2015) [PubMed] Article
More Info.:
Target
Name:
Thiol:disulfide interchange protein DsbA
Synonyms:
DSBA_ECOLI | JW3832 | Thiol:disulfide interchange protein DsbA | dsbA | dsf | dsf | ppfA
Type:
PROTEIN
Mol. Mass.:
23103.76
Organism:
Escherichia coli (strain K12)
Description:
ChEMBL_109722
Residue:
208
Sequence:
MKKIWLALAGLVLAFSASAAQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEKK