Reaction Details
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Target
Sphingosine kinase 1
Ligand
BDBM50041978
Substrate
n/a
Meas. Tech.
ChEMBL_1582610 (CHEMBL3816951)
Ki
3.6±n/a nM
Citation
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More Info.:
Target
Name:
Sphingosine kinase 1
Synonyms:
SK 1 | SPHK1_MOUSE | SPK 1 | Sk1 | Sphk1
Type:
PROTEIN
Mol. Mass.:
42447.37
Organism:
Mus musculus
Description:
ChEMBL_107622
Residue:
382
Sequence:
MEPVECPRGLLPRPCRVLVLLNPQGGKGKALQLFQSRVQPFLEEAEITFKLILTERKNHARELVCAEELGHWDALAVMSGDGLMHEVVNGLMERPDWETAIQKPLCSLPGGSGNALAASVNHYAGYEQVTNEDLLINCTLLLCRRRLSPMNLLSLHTASGLRLYSVLSLSWGFVADVDLESEKYRRLGEIRFTVGTFFRLASLRIYQGQLAYLPVGTVASKRPASTLVQKGPVDTHLVPLEEPVPSHWTVVPEQDFVLVLVLLHTHLSSELFAAPMGRCEAGVMHLFYVRAGVSRAALLRLFLAMQKGKHMELDCPYLVHVPVVAFRLEPRSQRGVFSVDGELMVCEAVQGQVHPNYLWMVCGSRDAPSGRDSRRGPPPEEP