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Target
D(1A) dopamine receptor
Ligand
BDBM50019396
Substrate
n/a
Meas. Tech.
ChEMBL_58821 (CHEMBL668244)
Ki
4677±n/a nM
Citation
  TBA Bioorg Med Chem Lett 5:2371-2376 (1995)  
Target
Name:
D(1A) dopamine receptor
Synonyms:
DOPAMINE D1 | DRD1_RAT | Dopamine D1 high | Dopamine D1 low | Dopamine receptor | Dopamine receptor D1 | Dopamine1-like | Drd1 | Drd1a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49429.75
Organism:
RAT
Description:
P18901
Residue:
446
Sequence:
MAPNTSTMDEAGLPAERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPLGPFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLEDTEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKNCQTTAGNGNPVECAQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGSEETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIETVSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIAKPLEKLSPALSVILDYDTDVSLEKIQPVTHSGQHST
  
Inhibitor
Name:
BDBM50019396
Synonyms:
4-(2-Dipropylamino-ethyl)-benzene-1,2-diol | 4-(2-Dipropylamino-ethyl)-benzene-1,2-diol (N,N-dipropyldopamine) | CHEMBL15564 | N,N-di-n-Propyldopamine
Type:
Small organic molecule
Emp. Form.:
C14H23NO2
Mol. Mass.:
237.3379
SMILES:
CCCN(CCC)CCc1ccc(O)c(O)c1
Structure:
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