Reaction Details  Report a problem with these data
Target
5-hydroxytryptamine receptor 1A
Ligand
BDBM25761
Substrate
n/a
Ki
78±n/a nM
Comments
PDSP_1540
Citation
 Weber, JT; Hayataka, K; O'Connor, MF; Parker, KK Rabbit cerebral cortex 5HT1a receptors. Comp Biochem Physiol C, Pharmacol Toxicol Endocrinol 117:19-24 (1997) [PubMed]  Article
Target
Name:
5-hydroxytryptamine receptor 1A
Synonyms:
5-HT1A | HTR1A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
18528.48
Organism:
RABBIT
Description:
Q9MZ11
Residue:
170
Sequence:
IPPMLGWRTPEDRSDPDACTISKDHGYTIYSTFGAFYVPLLLMLVLYGRIFRAARFRIRKTVKKVEKKGADTRFGATPAPQPRKSVNGEPGSRDWRQGVENKGVGLACANGAVRQGDDGAALEVIEVHRVGNSKEHLPLPSEAGAASGAPASFERKNERNAEAKRKMALA
  
Inhibitor
Name:
BDBM25761
Synonyms:
Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-) | PROPRANOLOL, d | PROPRANOLOL, l- | PROPRANOLOL,(+) | PROPRANOLOL,(-) | Propanolol | Propanolol,(+/-) | Propranolol | [2-hydroxy-3-(naphthalen-1-yloxy)propyl](propan-2-yl)amine
Type:
Small organic molecule
Emp. Form.:
C16H21NO2
Mol. Mass.:
259.3434
SMILES:
CC(C)NCC(O)COc1cccc2ccccc12
Structure:
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