Reaction Details  Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM84738
Substrate
n/a
Ki
740±n/a nM
Comments
PDSP_813
Citation
 Setola, V; Hufeisen, SJ; Grande-Allen, KJ; Vesely, I; Glennon, RA; Blough, B; Rothman, RB; Roth, BL 3,4-methylenedioxymethamphetamine (MDMA, "Ecstasy") induces fenfluramine-like proliferative actions on human cardiac valvular interstitial cells in vitro. Mol Pharmacol 63:1223-9 (2003) [PubMed]  Article
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM84738
Synonyms:
CAS_16105-77-4 | Fenfluramine | Fenfluramine (+) | Fenfluramine (-) | NSC_3337 | d-Fenfluramine
Type:
Small organic molecule
Emp. Form.:
C12H16F3N
Mol. Mass.:
231.2573
SMILES:
CCNC(C)Cc1cccc(c1)C(F)(F)F
Structure:
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