Reaction Details  Report a problem with these data
Target
Promotilin
Ligand
BDBM86313
Substrate
n/a
Ki
190.55±n/a nM
Comments
PDSP_6110
Citation
 Dass, NB; Hill, J; Muir, A; Testa, T; Wise, A; Sanger, GJ The rabbit motilin receptor: molecular characterisation and pharmacology. Br J Pharmacol 140:948-54 (2003) [PubMed]  Article
Target
Name:
Promotilin
Synonyms:
MLN | MOTI_RABIT | Motilin | Promotilin
Type:
Enzyme Catalytic Domain
Mol. Mass.:
14668.99
Organism:
RABBIT
Description:
Motilin 0 RABBIT::P27114
Residue:
133
Sequence:
MVSRKAVAALLLVHVTAMLASQTEAFVPIFTYSELQRMQERERNRGHKKSLSVQQRSDAAAAPRPAEPTLEEENGRMQLTAPVEIGMRMNSRQLEKYRAALEAAERAVHPDAPSRPCWPAGGESGWSGEPSPT
  
Inhibitor
Name:
BDBM86313
Synonyms:
CAS_114-07-8 | NSC_12560 | erythromycin-A
Type:
Small organic molecule
Emp. Form.:
C37H67NO13
Mol. Mass.:
733.9268
SMILES:
CCC1OC(=O)C(C)C(OC2CC(C)(OC)C(O)C(C)O2)C(C)C(OC2OC(C)CC(C2O)N(C)C)C(C)(O)CC(C)C(=O)C(C)C(O)C1(C)O
Structure:
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