Reaction Details
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Target
Salicylate synthase
Ligand
BDBM92747
Substrate
n/a
Meas. Tech.
Fluorescence-Based Thermal Shift Assay
Ki
1.2e+4± 1e+3 nM
Citation
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More Info.:
Target
Name:
Salicylate synthase
Synonyms:
Isochorismate synthase/isochorismate-pyruvate lyase MbtI | MBTI_MYCTO | Salicylate synthase (MbtI) | mbtI | trpE2
Type:
Protein
Mol. Mass.:
48744.20
Organism:
Mycobacterium tuberculosis
Description:
P9WFX0
Residue:
450
Sequence:
MSELSVATGAVSTASSSIPMPAGVNPADLAAELAAVVTESVDEDYLLYECDGQWVLAAGVQAMVELDSDELRVIRDGVTRRQQWSGRPGAALGEAVDRLLLETDQAFGWVAFEFGVHRYGLQQRLAPHTPLARVFSPRTRIMVSEKEIRLFDAGIRHREAIDRLLATGVREVPQSRSVDVSDDPSGFRRRVAVAVDEIAAGRYHKVILSRCVEVPFAIDFPLTYRLGRRHNTPVRSFLLQLGGIRALGYSPELVTAVRADGVVITEPLAGTRALGRGPAIDRLARDDLESNSKEIVEHAISVRSSLEEITDIAEPGSAAVIDFMTVRERGSVQHLGSTIRARLDPSSDRMAALEALFPAVTASGIPKAAGVEAIFRLDECPRGLYSGAVVMLSADGGLDAALTLRAAYQVGGRTWLRAGAGIIEESEPEREFEETCEKLSTLTPYLVARQ