Reaction Details
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Target
Histone deacetylase 6 [440-798]
Ligand
BDBM25150
Substrate
n/a
Meas. Tech.
HDAC6 fluorescence anisotropy assay
Temperature
298.15±n/a K
Ki
1.1±0.2 nM
IC50
1.9±0.3 nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Histone deacetylase 6 [440-798]
Synonyms:
Catalytic domain 2 (zCD2) | zCD2
Type:
n/a
Mol. Mass.:
39850.25
Organism:
Danio rerio
Description:
F8W4B7[440-798]
Residue:
359
Sequence:
SSPITGLVYDQRMMLHHNMWDSHHPELPQRISRIFSRHEELRLLSRCHRIPARLATEEELALCHSSKHISIIKSSEHMKPRDLNRLGDEYNSIFISNESYTCALLAAGSCFNSAQAILTGQVRNAVAIVRPPGHHAEKDTACGFCFFNTAALTARYAQSITRESLRVLIVDWDVHHGNGTQHIFEEDDSVLYISLHRYEDGAFFPNSEDANYDKVGLGKGRGYNVNIPWNGGKMGDPEYMAAFHHLVMPIAREFAPELVLVSAGFDAARGDPLGGFQVTPEGYAHLTHQLMSLAAGRVLIILEGGYNLTSISESMSMCTSMLLGDSPPSLDHLTPLKTSATVSINNVLRAHAPFWSSLR