Reaction Details
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Target
Kappa-type opioid receptor [Q115A]
Ligand
BDBM214799
Substrate
n/a
Meas. Tech.
Homologous Competition Assay
pH
7.4±n/a
Temperature
298.15±n/a K
Ki
5.8e+2±2.8e+2 nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Kappa-type opioid receptor [Q115A]
Synonyms:
Kappa opioid receptor (KOR Q115A) | OPRK | OPRK1 | OPRK_HUMAN
Type:
Protein
Mol. Mass.:
42591.71
Organism:
Homo sapiens (Human)
Description:
Human KOR with Q115A mutation
Residue:
380
Sequence:
MDSPIQIFRGEPGPTCAPSACLPPNSSAWFPGWAEPDSNGSAGSEDAQLEPAHISPAIPVIITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFASTVYLMNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALGSTSHSTAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFPLKMRMERQSTSRVRNTVQDPAYLRDIDGMNKPV