Reaction Details
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Target
Kappa-type opioid receptor [Y139F]
Ligand
BDBM214799
Substrate
n/a
Meas. Tech.
cAMP Inhibition Assay
pH
7.4±n/a
EC50
1.4e+2±2e+1 nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Kappa-type opioid receptor [Y139F]
Synonyms:
Kappa opioid receptor (KOR Y139F) | OPRK | OPRK1 | OPRK_HUMAN
Type:
Protein
Mol. Mass.:
42632.76
Organism:
Homo sapiens (Human)
Description:
Human KOR with Y139F mutation
Residue:
380
Sequence:
MDSPIQIFRGEPGPTCAPSACLPPNSSAWFPGWAEPDSNGSAGSEDAQLEPAHISPAIPVIITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYLMNSWPFGDVLCKIVISIDFYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALGSTSHSTAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFPLKMRMERQSTSRVRNTVQDPAYLRDIDGMNKPV