Reaction Details Report a problem with these data
Target
Kappa-type opioid receptor [Y320F]
Ligand
BDBM214799
Substrate
n/a
Meas. Tech.
cAMP Inhibition Assay
pH
7.4±n/a
EC50
3e+2±5e+1 nM
Comments
extracted
Citation
Vardy, E; Mosier, PD; Frankowski, KJ; Wu, H; Katritch, V; Westkaemper, RB; Aubé, J; Stevens, RC; Roth, BL Chemotype-selective modes of action of ¿-opioid receptor agonists. J Biol Chem 288:34470-83 (2013) [PubMed] Article
More Info.:
Target
Name:
Kappa-type opioid receptor [Y320F]
Synonyms:
Kappa opioid receptor (KOR Y320F) | OPRK | OPRK1 | OPRK_HUMAN
Type:
Protein
Mol. Mass.:
42632.76
Organism:
Homo sapiens (Human)
Description:
Human KOR with Y320F mutation
Residue:
380
Sequence:
MDSPIQIFRGEPGPTCAPSACLPPNSSAWFPGWAEPDSNGSAGSEDAQLEPAHISPAIPVIITAVYSVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYLMNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALGSTSHSTAALSSYYFCIALGFTNSSLNPILYAFLDENFKRCFRDFCFPLKMRMERQSTSRVRNTVQDPAYLRDIDGMNKPV