Reaction Details
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Target
Bromodomain-containing protein 4 [352-457]
Ligand
BDBM220430
Substrate
n/a
Meas. Tech.
Bromodomain Domain Binding Assay
pH
6±n/a
Temperature
298.15±n/a K
Ki
4.2±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Bromodomain-containing protein 4 [352-457]
Synonyms:
BRD4 | BRD4_HUMAN | Bromodomain-containing protein 4 (BRD4) | Bromodomain-containing protein 4 (BRD4)(aa 352-457) | Bromodomain-containing protein 4 (BRD4-BD2) | HUNK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12432.37
Organism:
Homo sapiens (Human)
Description:
BDII: amino acid E352-M457
Residue:
106
Sequence:
EQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM