Reaction Details Report a problem with these data
Target
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
Ligand
BDBM50177715
Substrate
n/a
Meas. Tech.
ChEMBL_1581780 (CHEMBL3816306)
IC50
78±n/a nM
Citation
Hatcher, JM; Weisberg, E; Sim, T; Stone, RM; Liu, S; Griffin, JD; Gray, NS Discovery of a Highly Potent and Selective Indenoindolone Type 1 Pan-FLT3 Inhibitor. ACS Med Chem Lett 7:476-81 (2016) [PubMed] Article
More Info.:
Target
Name:
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
Synonyms:
PHKG | PHKG1 | PHKG1_HUMAN | Phosphorylase b kinase gamma catalytic chain, skeletal muscle isoform | Phosphorylase kinase | Phosphorylase kinase gamma subunit 1 | Phosphorylase kinase subunit gamma 1
Type:
PROTEIN
Mol. Mass.:
45025.22
Organism:
Homo sapiens (Human)
Description:
ChEMBL_774515
Residue:
387
Sequence:
MTRDEALPDSHSAQDFYENYEPKEILGRGVSSVVRRCIHKPTSQEYAVKVIDVTGGGSFSPEEVRELREATLKEVDILRKVSGHPNIIQLKDTYETNTFFFLVFDLMKRGELFDYLTEKVTLSEKETRKIMRALLEVICTLHKLNIVHRDLKPENILLDDNMNIKLTDFGFSCQLEPGERLREVCGTPSYLAPEIIECSMNEDHPGYGKEVDMWSTGVIMYTLLAGSPPFWHRKQMLMLRMIMSGNYQFGSPEWDDYSDTVKDLVSRFLVVQPQNRYTAEEALAHPFFQQYLVEEVRHFSPRGKFKVIALTVLASVRIYYQYRRVKPVTREIVIRDPYALRPLRRLIDAYAFRIYGHWVKKGQQQNRAALFENTPKAVLLSLAEEDY