Reaction Details Report a problem with these data
Target
Substance-K receptor
Ligand
BDBM50049750
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_218
Citation
Sullivan, JP; Donnelly-Roberts, D; Briggs, CA; Anderson, DJ; Gopalakrishnan, M; Piattoni-Kaplan, M; Campbell, JE; McKenna, DG; Molinari, E; Hettinger, AM; Garvey, DS; Wasicak, JT; Holladay, MW; Williams, M; Arneric, SP A-85380 [3-(2(S)-azetidinylmethoxy) pyridine]: in vitro pharmacological properties of a novel, high affinity alpha 4 beta 2 nicotinic acetylcholine receptor ligand. Neuropharmacology 35:725-34 (1996) [PubMed] Article
More Info.:
Target
Name:
Substance-K receptor
Synonyms:
NK-2 receptor | NK-2R | NK2R_BOVIN | Neurokinin 2 receptor | Neurokinin A receptor | SKR | Substance-K receptor | TAC2R | TACR2 | Tachykinin receptor 2
Type:
PROTEIN
Mol. Mass.:
43078.78
Organism:
Bos taurus
Description:
ChEMBL_143050
Residue:
384
Sequence:
MGACVVMTDINISSGLDSNATGITAFSMPGWQLALWTAAYLALVLVAVMGNATVIWIILAHQRMRTVTNYFIVNLALADLCMAAFNAAFNFVYASHNIWYFGRAFCYFQNLFPITAMFVSIYSMTAIAADRYMAIVHPFQPRLSAPGTRAVIAGIWLVALALAFPQCFYSTITTDEGATKCVVAWPEDSGGKMLLLYHLIVIALIYFLPLVVMFVAYSVIGLTLWRRSVPGHQAHGANLRHLQAKKKFVKTMVLVVVTFAICWLPYHLYFILGTFQEDIYCHKFIQQVYLALFWLAMSSTMYNPIIYCCLNHRFRSGFRLAFRCCPWVTPTEEDKMELTYTPSLSTRVNRCHTKEIFFMSGDVAPSEAVNGQAESPQAGVSTEP