Reaction Details Report a problem with these data
Target
Anthranilate phosphoribosyltransferase
Ligand
BDBM93073
Substrate
n/a
Meas. Tech.
Fluoresence-based Assay
Ki
1.5e+3± 1e+2 nM
Citation
Castell, A; Short, FL; Evans, GL; Cookson, TV; Bulloch, EM; Joseph, DD; Lee, CE; Parker, EJ; Baker, EN; Lott, JS The Substrate Capture Mechanism of Mycobacterium tuberculosis Anthranilate Phosphoribosyltransferase Provides a Mode for Inhibition. Biochemistry 52:1776-1787 (2013) [PubMed] Article
More Info.:
Target
Name:
Anthranilate phosphoribosyltransferase
Synonyms:
Anthranilate phosphoribosyltransferase (Mtb-AnPRT) | TRPD_MYCTO | trpD
Type:
Enzyme
Mol. Mass.:
37738.87
Organism:
Mycobacterium tuberculosis
Description:
P9WFX4
Residue:
370
Sequence:
MALSAEGSSGGSRGGSPKAEAASVPSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGGDGVNTVNLSTMAAIVVAAAGVPVVKHGNRAASSLSGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQI