Reaction Details Report a problem with these data
Target
Rhomboid-related protein 3
Ligand
BDBM50199883
Substrate
n/a
Meas. Tech.
Activity-based Protein Profiling (ABPP)
pH
7.4±0
Temperature
310.15±0 K
IC50
7.0e+4± 1.3e+4 nM
Citation
Wolf, EV; Zeissler, A; Verhelst, SH Inhibitor Fingerprinting of Rhomboid Proteases by Activity-Based Protein Profiling Reveals Inhibitor Selectivity and Rhomboid Autoprocessing. ACS Chem Biol 10:2325-33 (2015) [PubMed] Article
More Info.:
Target
Name:
Rhomboid-related protein 3
Synonyms:
RHBL3_MOUSE | Rhbdl3 | Rhbdl4 | Rhomboid protease (MmRHBDL3) | Rhomboid-related protein 3 | Vrho
Type:
Protein
Mol. Mass.:
45272.26
Organism:
Mus musculus (Mouse)
Description:
n/a
Residue:
404
Sequence:
MGEHPSPGPAVAACAEAERIEELEPEAEERLPAAPEDHWKVLFEKFDPGSTGYISTGKFRSLLESHSSKLDPHKKEVLLALADSHADGQICYQDFVNLMSNKRSNSFRQAILQGNRRLSSKALLEEKGLSLSQRLIRHVAYETLPREIDRKWYYDSYTCCPPPWFMITITLLEVALFLYNGVLLDQFVLQVTHPRYLKNSLVYHPQLRAQAWRYVTYIFMHAGVEQLGLNVALQLLVGVPLEMVHGATRIGLVYVAGVVAGSLAVSVADMTAPVVGSSGGVYALVSAHLANIVMNWSGMKCQFKLLRMAVALICMSMEFGRAVWLRFHPSAYPPCPHPSFVAHLGGVAVGITLGVVVLRNYEQRLQDQSLWWIFVTMYTIFVLFAVFWNIFAYTLLDLKLPPAP