Assay Method Information

Assay Name:  ChEMBL_2235877 (CHEMBL5149649)
Description:  Inhibition of N-terminal His-Smt-tagged MSK1 C-terminal kinase domain (414 to 738 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using FAM-PSKPAATRKRRWSAPESR-NH2 as substrate preincubated for 1 hr followed by substrate addition and measured after 70 mins by ADP-Glo kinase assay
Affinity data for this assay
 

If you find an error in this entry please send us an E-mail