Assay Method Information

Assay Name:  ChEMBL_1707632 (CHEMBL4058865)
Description:  Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by measuring URP pEC50 at 10'-5M preincubated for 15 mins followed by URP addition (Rvb = 8.09 +/- 0.03 No_unit)
Affinity data for this assay
 

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