Assay Method Information

Assay Name:  ChEMBL_1883064 (CHEMBL4384563)
Description:  Antagonist activity at human DEF3-fused CXCR4 receptor expressed in HEK293T cells co-expressing DAN1-HA-Galphaq/i5 assessed as inhibition of CXCL12-induced IP3 accumulation after 90 mins in presence of [3H]-myo-inositol by scintillation counting analysis
Affinity data for this assay
 

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