| Assay Method Information | |
| | ChEMBL_1883975 (CHEMBL4385474) |
| Description: | Antagonist activity at recombinant human N-terminal MDSKGSSQKGSRLLLLLVVSNLLLCQGVVS-tagged CXCR4 D187A mutant expressed in HEK293 cells assessed as inhibition of SDF1alpha-induced Gi activation preincubated for 30 mins followed by SDF1alpha addition and measured after 5 mins by BRET assay |
| Affinity data for this assay | |
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