Assay Method Information

Assay Name:  ChEMBL_2218663 (CHEMBL5131997)
Description:  Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells assessed as N-terminal biotinylated SRC1 box2 coactivator peptide recruitment by TR-FRET assay
Affinity data for this assay
 

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