Compile Data Set for Download or QSAR
Found 7 for UniProtKB: Q12913
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM231167(US9340574, 7)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0Assay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in 3,3-dimethylglutarate buffer (50 mM 3,3-dimethylglutarate, pH 7.0, 1 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9H4JUS Patent
LigandPNGBDBM81346(CHEMBL538798 | M9440 (Me-3,4-dephostatin))copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMT: 2°CAssay Description:In order to eliminated fluorescence interference, chemicals were subjected to a secondary screening using colorimetric BP incorporation assay. TGase...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2SZRPubMed
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM50544440(CHEMBL4647367 | US11192850, Entry 4t)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DEP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3R3BPubMed
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM50544431(CHEMBL4637459 | US11192850, Entry 4k)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DEP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3R3BPubMed
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM50544427(CHEMBL4632818 | US11192850, Entry 4g)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of DEP1 (unknown origin) expressed in Escherichia coli BL21 using p-nitrophenyl phosphate as substrate measured after 30 mins by UV-vis sp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3R3BPubMed
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM152210(US8987474, NSC-87877)copy SMILEScopy InChI
Affinity DataIC50: 6.56E+4nMAssay Description:NSC-87877 ranked among top 10% (175th) of the compounds with the best GLIDE scores for the docking to the human Shp2 PTP domain in our virtual screen...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZS2V61US Patent
TargetReceptor-type tyrosine-protein phosphatase eta(Homo sapiens (Human))
Indiana University Research and Technology Corporation

US Patent
LigandPNGBDBM50071058((2R,4aS,6aS,12bR,14aS,14bR)-10-Hydroxy-2,4a,6a,9,1...)copy SMILEScopy InChI
Affinity DataIC50: 1.12E+5nMAssay Description:Inhibition of human PTPRJ (1019 to 1311 residues) expressed in Escherichia coli strain BL21(DE3) using DiFMUP as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44TN9PubMed