Affinity DataIC50: 630nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 630nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 880nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 2.37E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 2.57E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 3.02E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 3.29E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 3.54E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 3.87E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 5.45E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 5.45E+3nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 7.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 8.13E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataEC50: 646nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 347nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 646nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 209nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 81nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 83nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
