Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554781 (CHEMBL4749280) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554782 (CHEMBL4783937) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554786 (CHEMBL4745076) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554780 (CHEMBL4791793) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554787 (CHEMBL4752328) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554784 (CHEMBL4759130) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554785 (CHEMBL4763851) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554789 (CHEMBL4758729) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554788 (CHEMBL4744468) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dedicator of cytokinesis protein 5 (Homo sapiens) | BDBM50554783 (CHEMBL4795607) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01201 BindingDB Entry DOI: 10.7270/Q2V40ZVJ | |||||||||||
More data for this Ligand-Target Pair |