BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 10 hits of affinity data for UniProtKB/TrEMBL: Q9H7D0   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554781
PNG
(CHEMBL4749280)
Show SMILES COc1ccc(cc1C)N1CCC2(CCN(Cc3cccc(Cl)c3)C2)C1=O
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 8.00E+3n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554782
PNG
(CHEMBL4783937)
Show SMILES Fc1cccc(c1)N1CCC2(CCN(Cc3cccc(Cl)c3)C2)C1=O
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554786
PNG
(CHEMBL4745076)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2cnc3ccccc3c2)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.20E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554780
PNG
(CHEMBL4791793)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2cccc(Cl)c2)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.40E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554787
PNG
(CHEMBL4752328)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2ccc(Cl)c(Cl)c2)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.90E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554784
PNG
(CHEMBL4759130)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2ccc3CCCc3c2)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.20E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554785
PNG
(CHEMBL4763851)
Show SMILES Cn1cc(CN2CC[C@@]3(C2)[C@@H](O)CN(c2ccccc2)S3(=O)=O)c2ccccc12 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.30E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554789
PNG
(CHEMBL4758729)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2ccccc2Cl)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.50E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554788
PNG
(CHEMBL4744468)
Show SMILES O[C@H]1CN(c2ccccc2)S(=O)(=O)[C@@]11CCN(Cc2ccc(Cl)cc2)C1 |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.60E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair
Dedicator of cytokinesis protein 5


(Homo sapiens)
BDBM50554783
PNG
(CHEMBL4795607)
Show SMILES COc1ccc(CN2CC[C@@]3(C2)[C@@H](O)CN(c2ccccc2)S3(=O)=O)cc1F |r|
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 4.40E+4n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of N-terminal GFP tagged human DOCK5 (1212-1642 residues) expressed in HEK293T cells assessed as reduction in exchange activity incubated ...


Citation and Details

Article DOI: 10.1021/acs.jmedchem.0c01201
BindingDB Entry DOI: 10.7270/Q2V40ZVJ
More data for this
Ligand-Target Pair