23 articles for thisTarget

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The following articles (labelled with PubMed ID or TBD) are for your review

PMID	Data	Article Title	Organization
24900877	107	Development of novel benzomorpholine class of diacylglycerol acyltransferase I inhibitors.	Merck Research Laboratories
24618302	49	Discovery of novel quinoline carboxylic acid series as DGAT1 inhibitors.	Merck Research Laboratories
24670009	65	Discovery of 6-phenylpyrimido[4,5-b][1,4]oxazines as potent and selective acyl CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitors with in vivo efficacy in rodents.	Amgen
23711919	62	Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 3.	Kitasato University
23665143	8	Manzamine A, a marine-derived alkaloid, inhibits accumulation of cholesterol ester in macrophages and suppresses hyperlipidemia and atherosclerosis in vivo.	Kumamoto University
23535327	44	Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 2.	Kitasato University
23369538	88	Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 1.	Kitasato University
23317570	42	Lead optimization of a pyridine-carboxamide series as DGAT-1 inhibitors.	Merck Research Laboratories
23116186	68	Design and optimization of pyrazinecarboxamide-based inhibitors of diacylglycerol acyltransferase 1 (DGAT1) leading to a clinical candidate dimethylpyrazinecarboxamide phenylcyclohexylacetic acid (AZD7687).	Astrazeneca
18284184	4	Biphenyl versus phenylpyridazine derivatives: the role of the heterocycle in a series of acyl-CoA:cholesterol acyl transferase inhibitors.	Universita Di Milano
21413799	63	Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the potential treatment of obesity and diabetes.	Hoffmann-La Roche
17157006	21	Human ACAT inhibitory effects of shikonin derivatives from Lithospermum erythrorhizon.	National Research Laboratory of Lipid Metabolism and Atherosclerosis
16919944	25	Anti-atherosclerotic and anti-inflammatory activities of catecholic xanthones and flavonoids isolated from Cudrania tricuspidata.	National Research Laboratory of Lipid Metabolism and Atherosclerosis
16302810	9	Mono- or diphenylpyridazines connected to N-(2,4-difluorophenyl)-N'-heptylurea as acyl-CoA:cholesterol acyltransferase inhibitors.	Università
15603959	12	Saucerneol B derivatives as human acyl-CoA: cholesterol acyltransferase inhibitors.	Korea Research Institute of Bioscience and Biotechnology
15324887	2	Synthesis of cinnamic acid derivatives and their inhibitory effects on LDL-oxidation, acyl-CoA:cholesterol acyltransferase-1 and -2 activity, and decrease of HDL-particle size.	National Research Laboratory of Lipid Metabolism and Atherosclerosis
15149654	7	Human ACAT-1 and -2 inhibitory activities of saucerneol B, manassantin A and B isolated from Saururus chinensis.	Korea Research Institute of Bioscience and Biotechnology
32035699	8	Inhibition of cholesteryl ester synthesis by polyacetylenes from Atractylodes rhizome.	Kitasato University
30433781	23	Discovery of Clinical Candidate 2-(4-(2-((1 H-Benzo[ d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)- N-(6-methyl-2,4-bis(methylthio)pyridin-3-yl)acetamide Hydrochloride [K-604], an Aqueous-Soluble Acyl-CoA:Cholesterol O-Acyltransferase-1 Inhibitor.	Kowa
29456796	51	Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1.	Glaxosmithkline
28242547	2	Vicinal diaryl azole-based urea derivatives as potential cholesterol lowering agents acting through inhibition of SOAT enzymes.	The Maharaja Sayajirao University of Baroda
19152636	26	Probing the active site of Candida glabrata dihydrofolate reductase with high resolution crystal structures and the synthesis of new inhibitors.	University of Connecticut