The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27654218 |
56 |
Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors. |
Ludwig-Maximilians-Universit£T M£Nchen |
25147609 |
18 |
Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor. |
Hokkaido University |
25698617 |
61 |
Design, synthesis and SAR studies of GABA uptake inhibitors derived from 2-substituted pyrrolidine-2-yl-acetic acids. |
Ludwig-Maximilians-Universit£T M£Nchen |
24112084 |
6 |
The lignan (-)-hinokinin displays modulatory effects on human monoamine and GABA transporter activities. |
Drexel University College of Medicine |
23886812 |
16 |
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports. |
Hokkaido University |
23770450 |
3 |
Synthesis of N-substituted acyclicß-amino acids and their investigation as GABA uptake inhibitors. |
Zentrum F£R Pharmaforschung |
21940173 |
32 |
Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation. |
Ludwig-Maximilians-University Munich |
16246548 |
22 |
Design, synthesis, and biological evaluation of the N-diarylalkenyl-piperidinecarboxylic acid derivatives as GABA uptake inhibitors (I). |
Fudan University |
21353350 |
61 |
Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors. |
Ludwig-Maximilians-University Munich |
21134748 |
59 |
Stereospecific synthesis and structure-activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors. |
Glaxosmithkline |
20219271 |
10 |
Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship. |
Zentrum F£R Pharmaforschung |
| 20 |
On the bioactive conformation of the gaba uptake inhibitor SK&F 89976-A |
TBA |
30777661 |
42 |
Screening oxime libraries by means of mass spectrometry (MS) binding assays: Identification of new highly potent inhibitors to optimized inhibitors ?-aminobutyric acid transporter 1. |
Ludwig-Maximilians-University M£Nchen |
31117514 |
167 |
Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at ?-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters. |
University of Copenhagen |
30376325 |
50 |
Novel Allosteric Ligands of ?-Aminobutyric Acid Transporter 1 (GAT1) by MS Based Screening of Pseudostatic Hydrazone Libraries. |
Ludwig-Maximilians-Universit£T M£Nchen |
8057281 |
100 |
Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3. |
Synaptic Pharmaceutical |
28991462 |
360 |
Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/?-Aminobutyric Acid Transporter 1 (BGT1). |
University of Copenhagen |