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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
3336036 83 New potent antagonists of leukotrienes C4 and D4. 1. Synthesis and structure-activity relationships.EBI Ono Pharmaceutical
3027332 18 Substituted (aryloxy)alkanoic acids as antagonists of slow-reacting substance of anaphylaxis.EBI TBA
3016267 46 Synthesis and structure-activity relationship studies of a series of 5-aryl-4,6-dithianonanedioic acids and related compounds: a novel class of leukotriene antagonists.EBI TBA
9873435 10 Development of new chromanol antagonists of leukotriene D4.EBI Pfizer
26985325 62 Discovery of 3-Substituted 1H-Indole-2-carboxylic Acid Derivatives as a Novel Class of CysLT1 Selective Antagonists.EBI Shanghai Institute of Materia Medica
26200813 90 Discovery of Gemilukast (ONO-6950), a Dual CysLT1 and CysLT2 Antagonist As a Therapeutic Agent for Asthma.EBI Setsunan University
25800431 30 Discovery of a potent, orally available dual CysLT1 and CysLT2 antagonist with dicarboxylic acid.EBI Ono Pharmaceutical
25408836 44 Discovery of Highly Potent Dual CysLT1 and CysLT2 Antagonist.EBI Ono Pharmaceutical
3033245 28 Leukotriene receptor antagonists. 2. The [[(tetrazol-5-ylaryl)oxy]methyl]acetophenone derivatives.EBI TBA
1331447 32 Development of a novel series of styrylquinoline compounds as high-affinity leukotriene D4 receptor antagonists: synthetic and structure-activity studies leading to the discovery of (+-)-3-[[[3-[2-(7-chloro-2-quinolinyl)-(E)-ethenyl]phenyl][[3- (dimethylamino)-3-oxopropyl]thio]methyl]thio]propionicEBI Merck Frosst Centre For Therapeutic Research
9871597 65 A series of non-quinoline cysLT1 receptor antagonists: SAR study on pyridyl analogs of Singulair.EBI Merck Frosst Center For Therapeutic Research
9871521 32 Synthesis and SAR of a novel, potent and structurally simple LTD4 antagonist of the quinoline class.EBI Novartis Pharma
30613325 88 Discovery of Orally Bioavailable and Liver-Targeted Hypoxia-Inducible Factor Prolyl Hydroxylase (HIF-PHD) Inhibitors for the Treatment of Anemia.EBI Merck
23455026 2 Structure-based drug design using GPCR homology modeling: toward the discovery of novel selective CysLT2 antagonists.EBI Zhejiang University
9089329 48 Synthesis and structure-activity relationships of carboxylated chalcones: a novel series of CysLT1 (LTD4) receptor antagonists.EBI Vrije Universiteit
2547071 27 3,4-Dihydro-2H-1-benzopyran-2-carboxylic acids and related compounds as leukotriene antagonists.EBI Roche Research Center
2342072 46 Evolution of a series of peptidoleukotriene antagonists: synthesis and structure/activity relationships of 1,3,5-substituted indoles and indazoles.EBI Ici Pharmaceuticals Group
2170649 37 The development of a novel series of (quinolin-2-ylmethoxy)phenyl-containing compounds as high-affinity leukotriene receptor antagonists. 3. Structural variation of the acidic side chain to give antagonists of enhanced potency.EBI Rorer Central Research
2157009 49 Development of a novel series of (2-quinolinylmethoxy)phenyl-containing compounds as high-affinity leukotriene receptor antagonists. 1. Initial structure-activity relationships.EBI Rorer Central Research