The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28186757 |
66 |
Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 2: Structure-Based Drug Design and Structure-Activity Relationship.![EBI](/images/logo_chembl.png) |
European Institute of Oncology |
28186755 |
85 |
Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration.![EBI](/images/logo_chembl.png) |
European Institute of Oncology |
28065500 |
8 |
Activation of lysine-specific demethylase 1 inhibitor peptide by redox-controlled cleavage of a traceless linker.![EBI](/images/logo_chembl.png) |
Nagoya City University |
26702542 |
59 |
Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent.![EBI](/images/logo_chembl.png) |
European Institute of Oncology |
24883177 |
10 |
Synthesis and evaluation of novel cyclic Peptide inhibitors of lysine-specific demethylase 1.![EBI](/images/logo_chembl.png) |
Medical University of South Carolina |
25580204 |
10 |
3,5-Diamino-1,2,4-triazoles as a novel scaffold for potent, reversible LSD1 (KDM1A) inhibitors.![EBI](/images/logo_chembl.png) |
Medical University of South Carolina |
25585008 |
28 |
Further insights into the SAR of ?-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A.![EBI](/images/logo_chembl.png) |
University of Parma |
29459279 |
10 |
Cyclic peptide inhibitors of lysine-specific demethylase 1 with improved potency identified by alanine scanning mutagenesis.![EBI](/images/logo_chembl.png) |
Medical University of South Carolina |