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11 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
23562062 4 Arylsulfonamide pyrimidines as VLA-4 antagonists.EBI Elan Pharmaceuticals
15214773 76 Fragment-based drug discovery.EBI Sunesis Pharmaceuticals
12139455 78 Selective alpha4beta7 integrin antagonists and their potential as antiinflammatory agents.EBI Genentech
21109434 40 Structure-activity relationship (SAR) of thea-amino acid residue of potent tetrahydroisoquinoline (THIQ)-derived LFA-1/ICAM-1 antagonists.EBI Sunesis Pharmaceuticals
15686933 12 De novo design, synthesis, and in vitro activity of LFA-1 antagonists based on a bicyclic[5.5]hydantoin scaffold.EBI Cerep
15481974 43 Second-generation lymphocyte function-associated antigen-1 inhibitors: 1H-imidazo[1,2-alpha]imidazol-2-one derivatives.EBI Boehringer Ingelheim Pharmaceuticals
11728185 55 Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 4. Structure-activity relationship of substituents on the benzene ring of the cinnamide.EBI Abbott Laboratories
11312920 23 Novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intracellular adhesion molecule-1 interaction. 2. Mechanism of inhibition and structure-based improvement of pharmaceutical properties.EBI Abbott Laboratories
31999923 16 Insights into Protein-Ligand Interactions in Integrin Complexes: Advances in Structure Determinations.EBI Pliant Therapeutics
7707308 3 Novel thiazole based heterocycles as inhibitors of LFA-1/ICAM-1 mediated cell adhesion.EBI R. W. Johnson Pharmaceutical Research Institute