The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27692854 |
100 |
N-Arylsulfonyl-a-amino carboxamides are potent and selective inhibitors of the chemokine receptor CCR10 that show efficacy in the murine DNFB model of contact hypersensitivity. |
Boehringer Ingelheim Pharmaceuticals |
22650618 |
4 |
Rediocide A, an Insecticide, induces G-protein-coupled receptor desensitization via activation of conventional protein kinase C. |
Chinese Academy of Sciences |
16198561 |
99 |
Novel CCR1 antagonists with oral activity in the mouse collagen induced arthritis. |
Novartis Institutes For Biomedical Research |
19674898 |
31 |
Spiropiperidine CCR5 antagonists. |
Roche Palo Alto |
19014885 |
32 |
Discovery of a potent, selective and orally bioavailable 3,9-diazaspiro[5.5]undeca-2-one CCR5 antagonist. |
Roche Palo Alto |
31882297 |
129 |
Discovery of small molecule antagonists of chemokine receptor CXCR6 that arrest tumor growth in SK-HEP-1 mouse xenografts as a model of hepatocellular carcinoma. |
Sanford Burnham Prebys Medical Discovery Institute |
30098865 |
60 |
Identification of a novel series of potent and selective CCR6 inhibitors as biological probes. |
Takeda Pharmaceutical |
29406702 |
128 |
Discovery of Novel 1-Cyclopentenyl-3-phenylureas as Selective, Brain Penetrant, and Orally Bioavailable CXCR2 Antagonists. |
Gsk Pharmaceuticals R & D |
25290020 |
4 |
n-Alkylboronic acid inhibitors reveal determinants of ligand specificity in the quorum-quenching and siderophore biosynthetic enzyme PvdQ. |
The University of Texas |
24977643 |
9 |
Broad-spectrum allosteric inhibition of herpesvirus proteases. |
University of California San Francisco |
16950396 |
13 |
Quantitative evaluation of each catalytic subsite of cathepsin B for inhibitory activity based on inhibitory activity-binding mode relationship of epoxysuccinyl inhibitors by X-ray crystal structure analyses of complexes. |
Osaka University of Pharmaceutical Sciences |