43 articles for thisTarget

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The following articles (labelled with PubMed ID or TBD) are for your review

PMID	Data	Article Title	Organization
10915041	2	Synthesis of fluorescent probes directed to the active site gorge of acetylcholinesterase.	The University of Montana
27908752	55	N-Propargylpiperidines with naphthalene-2-carboxamide or naphthalene-2-sulfonamide moieties: Potential multifunctional anti-Alzheimer's agents.	University of Ljubljana
27448914	30	Ameliorative effects of amide derivatives of 1,3,4-thiadiazoles on scopolamine induced cognitive dysfunction.	University Institute of Pharmaceutical Sciences
27598521	22	Discovery of Selective Inhibitors Targeting Acetylcholinesterase 1 from Disease-Transmitting Mosquitoes.	Ume£
26116179	5	Structure-based development of nitroxoline derivatives as potential multifunctional anti-Alzheimer agents.	University of Ljubljana
25468034	33	Synthesis of aminoalkyl-substituted aurone derivatives as acetylcholinesterase inhibitors.	Kyung Hee University
25226236	19	Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor.	University of Ljubljana
24485122	9	Synthesis of aminoalkyl-substituted coumarin derivatives as acetylcholinesterase inhibitors.	Kyung Hee University
23984975	29	Divergent structure-activity relationships of structurally similar acetylcholinesterase inhibitors.	Ume£
23941108	1	Casuarinines A-J, lycodine-type alkaloids from Lycopodiastrum casuarinoides.	Fudan University
8558505	77	A comparative molecular field analysis study of N-benzylpiperidines as acetylcholinesterase inhibitors.	University of Missouri St. Louis
23026084	17	Lead optimization studies towards the discovery of novel carbamates as potent AChE inhibitors for the potential treatment of Alzheimer's disease.	Csir-Central Drug Research Institute
18479118	114	Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.	Universit£
18333606	29	Bis-(-)-nor-meptazinols as novel nanomolar cholinesterase inhibitors with high inhibitory potency on amyloid-beta aggregation.	Fudan University
15214773	76	Fragment-based drug discovery.	Sunesis Pharmaceuticals
7490731	45	Synthesis and structure-activity relationships of acetylcholinesterase inhibitors: 1-benzyl-4-[(5,6-dimethoxy-1-oxoindan-2-yl)methyl]piperidine hydrochloride and related compounds.	Eisai
1552502	74	Synthesis and cholinergic properties of bis[[(dimethylamino)methyl]furanyl] analogues of ranitidine.	University of South Carolina
18438404	13	Activation of the endocannabinoid system by organophosphorus nerve agents.	University of California
20137941	44	Design, synthesis and evaluation of carbamate-modified (-)-N(1)-phenethylnorphysostigmine derivatives as selective butyrylcholinesterase inhibitors.	Kyoto University
20137934	38	Design, synthesis, evaluation and QSAR analysis of N(1)-substituted norcymserine derivatives as selective butyrylcholinesterase inhibitors.	Kyoto University
	27	Synthesis and anti-acetylcholinesterase activity of 1-benzyl-4-[(5,6-dimethoxy-1-indanon-2-yl)methyl]piperidine hydrochloride (E2020) and related compounds	TBA
30822710	39	Design, synthesis, and evaluation of isoflavone analogs as multifunctional agents for the treatment of Alzheimer's disease.	Chinese Academy of Medical Sciences and Peking Union Medical College
27519464	18	Coumarin derivatives as potential inhibitors of acetylcholinesterase: Synthesis, molecular docking and biological studies.	Panjab University
31078410	5	A new lateral root growth inhibitor from the sponge-derived fungus Aspergillus sp. LS45.	Ningbo University
30744931	170	Anti-cholinesterase hybrids as multi-target-directed ligands against Alzheimer's disease (1998-2018).	Csir-Central Drug Research Institute
31609115	50	Highly Selective Butyrylcholinesterase Inhibitors with Tunable Duration of Action by Chemical Modification of Transferable Carbamate Units Exhibit Pronounced Neuroprotective Effect in an Alzheimer's Disease Mouse Model.	Julius Maximilian University W£Rzburg
31082225	26	Rational Design of Multitarget-Directed Ligands: Strategies and Emerging Paradigms.	China Pharmaceutical University
30578075	14	In silico, NMR and pharmacological evaluation of an hydroxyoxindole cholinesterase inhibitor.	Universidade De £Vora
8709135	20	Identification of a 3-hydroxylated tacrine metabolite in rat and man: metabolic profiling implications and pharmacology.	Warner-Lambert
8027982	19	Syntheses and anticholinesterase activity of tetrahydrobenzazepine carbamates.	Pfizer
30340901	22	Design, synthesis, cholinesterase inhibition and molecular modelling study of novel tacrine hybrids with carbohydrate derivatives.	Universidade Federal Do Rio Grande Do Sul
29873484	25	Druggability Assessment of Targets Used in Kinetic Target-Guided Synthesis.	University of Groningen
29195794	12	Design, synthesis and pharmacological evaluation of some novel indanone derivatives as acetylcholinesterase inhibitors for the management of cognitive dysfunction.	Panjab University
29227101	30	The Magic of Crystal Structure-Based Inhibitor Optimization: Development of a Butyrylcholinesterase Inhibitor with Picomolar Affinity and in Vivo Activity.	University of Ljubljana
1469686	53	Synthesis and structure-activity relationships of acetylcholinesterase inhibitors: 1-benzyl-4-(2-phthalimidoethyl)piperidine and related derivatives.	Eisai
20846091	3	A FLT3-inhibitory constituent from the rhizomes of Anemarrhena asphodeloides.	Gyeongsang National University
14718605	8	Identification and characterization of 4-[[4-(2-butynyloxy)phenyl]sulfonyl]-N-hydroxy-2,2-dimethyl-(3S)thiomorpholinecarboxamide (TMI-1), a novel dual tumor necrosis factor-alpha-converting enzyme/matrix metalloprotease inhibitor for the treatment of rheumatoid arthritis.	Wyeth Research