The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27818110 |
61 |
Discovery of highly potent and selective orexin 1 receptor antagonists (1-SORAs) suitable for in vivo interrogation of orexin 1 receptor pharmacology. |
Merck Research Laboratories |
21831639 |
32 |
Discovery process and pharmacological characterization of a novel dual orexin 1 and orexin 2 receptor antagonist useful for treatment of sleep disorders. |
Glaxosmithkline |
24737316 |
18 |
Structural basis of pharmacological chaperoning for human ß-galactosidase. |
The University of Tokyo |
11809867 |
38 |
A(3) adenosine receptors in human neutrophils and promyelocytic HL60 cells: a pharmacological and biochemical study. |
University of Ferrara |
12573694 |
13 |
Pin1 and Par14 peptidyl prolyl isomerase inhibitors block cell proliferation. |
Tohoku University |
19054673 |
66 |
5,6-Dihydro-1H-pyridin-2-ones as potent inhibitors of HCV NS5B polymerase. |
Anadys Pharmaceuticals |
19267475 |
118 |
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins. |
Sapienza University of Rome |
18620380 |
8 |
Selectivity determinants of inhibitor binding to human 20alpha-hydroxysteroid dehydrogenase: crystal structure of the enzyme in ternary complex with coenzyme and the potent inhibitor 3,5-dichlorosalicylic acid. |
Monash University |
18579385 |
132 |
Carbonic anhydrase inhibitors: inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid. |
Universita Degli Studi Di Firenze |
18621524 |
17 |
The identification of potent, selective and CNS penetrant furan-based inhibitors of B-Raf kinase. |
Gsk |
8464047 |
14 |
Cyclic sulfolanes as novel and high affinity P2 ligands for HIV-1 protease inhibitors. |
Merck Research Laboratories |