The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26710088 |
248 |
Recent Progress in Histone Demethylase Inhibitors. |
University of Oxford |
26699912 |
108 |
Docking and Linking of Fragments To Discover Jumonji Histone Demethylase Inhibitors. |
University of Oxford |
26741168 |
239 |
8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors. |
The Institute of Cancer Research |
23964788 |
56 |
Identification of the KDM2/7 histone lysine demethylase subfamily inhibitor and its antiproliferative activity. |
Kyoto Prefectural University of Medicine |
23725560 |
22 |
Quantitative analysis of histone demethylase probes using fluorescence polarization. |
University of Colorado |
22724510 |
84 |
Plant growth regulator daminozide is a selective inhibitor of human KDM2/7 histone demethylases. |
University of Oxford |
21955276 |
60 |
Lysine demethylases inhibitors. |
Kyoto Prefectural University of Medicine |
32551003 |
53 |
Design and Synthesis of Styrenylcyclopropylamine LSD1 Inhibitors. |
Constellation Pharmaceuticals |
30745098 |
24 |
Identification of novel lysine demethylase 5-selective inhibitors by inhibitor-based fragment merging strategy. |
Kyoto Prefectural University of Medicine |
31158747 |
257 |
C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays. |
Institute of Cancer Research |
26682034 |
229 |
Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor. |
University of Oxford |
24325601 |
74 |
Pan-histone demethylase inhibitors simultaneously targeting Jumonji C and lysine-specific demethylases display high anticancer activities. |
Sapienza University of Rome |
29627262 |
109 |
Structure-based design and discovery of potent and selective KDM5 inhibitors. |
Celgene |
28160945 |
12 |
In search of new a-glucosidase inhibitors: Imidazolylpyrazole derivatives. |
University of The Punjab |
19217287 |
30 |
Development of multitargeted inhibitors of both the insulin-like growth factor receptor (IGF-IR) and members of the epidermal growth factor family of receptor tyrosine kinases. |
Abbott Laboratories |
12419810 |
6 |
Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight. |
University of Padova |