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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
16644215 52 Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors.EBI Celera Genomics
16554154 9 Development of activity-based probes for trypsin-family serine proteases.EBI Celera Genomics
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University of Florida
12930148 41 Potent, small-molecule inhibitors of human mast cell tryptase. Antiasthmatic action of a dipeptide-based transition-state analogue containing a benzothiazole ketone.EBI Johnson & Johnson Pharmaceutical Research & Development
16725321 13 Novel, potent, selective, and orally bioavailable human betaII-tryptase inhibitors.EBI Celera Genomics
15911249 29 Design, synthesis, and biological activity of potent and selective inhibitors of mast cell tryptase.EBI Aventis Pharmaceuticals
15745817 14 Combinatorial approaches towards the discovery of new tryptase inhibitors.EBI University of Barcelona
15546728 15 Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human beta-tryptase.EBI Aventis Pharmaceuticals
15341931 15 Novel pyrazinone inhibitors of mast cell tryptase: synthesis and SAR evaluation.EBI Aventis Pharmaceuticals
11959009 7 Bivalent inhibition of beta-tryptase: distance scan of neighboring subunits by dibasic inhibitors.EBI Institut FüR Biochemie
11527724 30 Monocharged inhibitors of mast cell tryptase derived from potent and selective dibasic inhibitors.EBI Axys Pharmaceuticals
11055355 72 Dibasic inhibitors of human mast cell tryptase. Part 1: synthesis and optimization of a novel class of inhibitors.EBI Axys Pharmaceuticals
27563406 128 Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B (Autophagin-1) Inhibitors.EBI Roche Pharma Research and Early Development
30995036 52 Design, Synthesis, and Preclinical Characterization of Selective Factor D Inhibitors Targeting the Alternative Complement Pathway.EBI Novartis Institutes For Biomedical Research