The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
11459661 |
41 |
Synthesis of N(1)-substituted analogues of (2R,4R)-4-amino-pyrrolidine-2,4-dicarboxylic acid as agonists, partial agonists, and antagonists of group II metabotropic glutamate receptors. |
Georgetown University Medical Center |
11412983 |
9 |
New probes of the agonist binding site of metabotropic glutamate receptors. |
Universit£ |
10397508 |
8 |
1-amino-APDC, a partial agonist of group II metabotropic glutamate receptors with neuroprotective properties. |
Georgetown University Medical Center |
| 6 |
Synthesis and biological activity of cyclic analogues of MPPG and MCPG as metabotropic glutamate receptor antagonists |
TBA |
| 15 |
Synthesis, molecular modeling, and biology of the 1-benzyl derivative of APDC-an apparent mGluR6 selective ligand |
TBA |
32173198 |
58 |
Discovery of 4-arylquinoline-2-carboxamides, highly potent and selective class of mGluR2 negative allosteric modulators: From HTS to activity in animal models. |
Merck |
10386938 |
16 |
Structure-activity relationships of substituted 5H-thiazolo[3,2-a]pyrimidines as group 2 metabotropic glutamate receptor antagonists. |
F. Hoffmann-La Roche |
9873635 |
67 |
2,3'-disubstituted-2-(2'-carboxycyclopropyl)glycines as potent and selective antagonists of metabotropic glutamate receptors. |
Eli Lilly |
30350962 |
102 |
Discovery of Novel Central Nervous System Penetrant Metabotropic Glutamate Receptor Subtype 2 (mGlu |
Vanderbilt University School of Medicine |
8632404 |
3 |
(2S,4S)-2-amino-4-(4,4-diphenylbut-1-yl)- pentane-1,5-dioic acid: a potent and selective antagonist for metabotropic glutamate receptors negatively linked to adenylate cyclase. |
Centre De Neurochimie Du Cnrs |
30146095 |
12 |
Amelioration of PXR-mediated CYP3A4 induction by mGluR2 modulators. |
Sanofi Us |
29057060 |
100 |
Discovery of VU6005649, a CNS Penetrant mGlu |
Vanderbilt University |
8813606 |
15 |
[3H]5-hydroxytryptamine labels the agonist high affinity state of the cloned rat 5-HT4 receptor. |
Synaptic Pharmaceutical |