The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27526040 |
21 |
Design and synthesis of new potent PTP1B inhibitors with the skeleton of 2-substituted imino-3-substituted-5-heteroarylidene-1,3-thiazolidine-4-one: Part I. |
Xi'An Jiaotong University |
| 25938987 |
49 |
Is RK-682 a promiscuous enzyme inhibitor? Synthesis and in vitro evaluation of protein tyrosine phosphatase inhibition of racemic RK-682 and analogues. |
University of Campinas |
| 25703307 |
30 |
Synthesis and biological evaluation of 3-aminoisoquinolin-1(2H)-one based inhibitors of the dual-specificity phosphatase Cdc25B. |
University of Pittsburgh |
| 25124112 |
54 |
Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors. |
Liaoning Normal University |
| 25497963 |
19 |
Bioactive constituents from the green alga Caulerpa racemosa. |
Nanchang University |
| 24090912 |
54 |
Design, synthesis, and biological evaluation of novel 2-ethyl-5-phenylthiazole-4-carboxamide derivatives as protein tyrosine phosphatase 1B inhibitors with improved cellular efficacy. |
Chinese Academy of Sciences |
| 23141909 |
46 |
Design and synthesis of novel bis-thiazolone derivatives as micromolar CDC25 phosphatase inhibitors: effect of dimerisation on phosphatase inhibition. |
University of Paris |
| 22506091 |
151 |
Dual-Specificity Phosphatase CDC25A/B Inhibitor Identified from a Focused Library with Nonelectrophilic Core Structure. |
TBA |
| 22705189 |
24 |
Arylstibonic acids are potent and isoform-selective inhibitors of Cdc25a and Cdc25b phosphatases. |
Imperial College |
| 22524450 |
24 |
Discovery of new inhibitors of Cdc25B dual specificity phosphatases by structure-based virtual screening. |
Universit£ |
| 18789703 |
14 |
Novel naphthoquinone and quinolinedione inhibitors of CDC25 phosphatase activity with antiproliferative properties. |
University of Paris |
| 11086732 |
10 |
Synthesis of the novel analogues of dysidiolide and their structure-activity relationship. |
The University of Tokyo |
| 21680062 |
77 |
Synthesis and biological evaluation of (±)-3-(2-(2-fluorobenzyloxy) naphthalen-6-yl)-2-aminopropanoic acid derivatives as novel PTP1B inhibitors. |
Yanbian University |
| 21665482 |
62 |
Facile fabrication of promising protein tyrosine phosphatase (PTP) inhibitor entities based on 'clicked' serine/threonine-monosaccharide hybrids. |
East China University of Science and Technology |
| 21420867 |
68 |
Using small molecules to target protein phosphatases. |
Max Planck Institute of Molecular Physiology |
| 21251827 |
60 |
A unique and rapid approach toward the efficient development of novel protein tyrosine phosphatase (PTP) inhibitors based on 'clicked' pseudo-glycopeptides. |
East China University of Science and Technology |
| 20363629 |
49 |
Discovery and structural optimization of pyrazole derivatives as novel inhibitors of Cdc25B. |
Chinese Academy of Sciences |
| 19969400 |
4 |
5-Substituted [1]pyrindine derivatives with antiproliferative activity. |
University of Paris |
| 19500977 |
20 |
Structure-based virtual screening approach to identify novel classes of Cdc25B phosphatase inhibitors. |
Sejong University |
| 19497739 |
66 |
Structure-based de novo design and biochemical evaluation of novel Cdc25 phosphatase inhibitors. |
Sejong University |
| 19028102 |
46 |
Bioactivities of simplified adociaquinone B and naphthoquinone derivatives against Cdc25B, MKP-1, and MKP-3 phosphatases. |
Virginia Polytechnic Institute and State University |
| 18714978 |
18 |
Discovery of novel Cdc25 phosphatase inhibitors with micromolar activity based on the structure-based virtual screening. |
Sejong University |
| 18334299 |
6 |
Tetramic and tetronic acids: an update on new derivatives and biological aspects. |
University of Bayreuth |
| 15497946 |
2 |
Marine sesquiterpenoids that inhibit the lyase activity of DNA polymerase beta. |
Virginia Polytechnic Institute and State University |
| 17379514 |
1 |
Fluorinated NSC as a Cdc25 inhibitor. |
Sejong University |
| 17084000 |
30 |
Synthesis and biological evaluation of dialkylsubstituted maleic anhydrides as novel inhibitors of Cdc25 dual specificity phosphatases. |
Université |
| 16434190 |
48 |
Synthesis of miltirone analogues as inhibitors of Cdc25 phosphatases. |
Graduate School of Chinese Academy of Sciences |
| 16289879 |
34 |
PTP-1B inhibitors: cyclopenta[d][1,2]-oxazine derivatives. |
Korea Research Institute of Chemical Technology |
| 15261298 |
23 |
Design and synthesis of novel Cdc25A-inhibitors having phosphate group as a hydrophilic residue. |
The University of Tokyo |
| 15149692 |
12 |
Design and synthesis of dysidiolide analogs from vitamin D3: novel class of Cdc25A inhibitors. |
The University of Tokyo |
| 15026048 |
30 |
Design and synthesis of macrocyclic inhibitors of phosphatase cdc25B. |
Schering |
| 12801222 |
76 |
Inhibition of Cdc25 phosphatases by indolyldihydroxyquinones. |
Duke University |
| 12113814 |
60 |
Synthesis and PTP1B inhibition of 1,2-naphthoquinone derivatives as potent anti-diabetic agents. |
Korea Research Institute of Chemical Technology |
| 11708908 |
55 |
Discovery and biological evaluation of a new family of potent inhibitors of the dual specificity protein phosphatase Cdc25. |
University of Pittsburgh |
| 11212099 |
107 |
Sulfonylated aminothiazoles as new small molecule inhibitors of protein phosphatases. |
University of Pittsburgh |
| 10762045 |
65 |
The solid phase synthesis of tetrahydroisoquinolines having cdc25B inhibitory activity. |
Pharmacia & Upjohn |
| 10498203 |
13 |
Dysidiolide and related gamma-hydroxy butenolide compounds as inhibitors of the protein tyrosine phosphatase, CDC25. |
Mitotix |
| 30978561 |
50 |
Synthesis and biological evaluation of tryptophan-derived rhodanine derivatives as PTP1B inhibitors and anti-bacterial agents. |
Yanbian University College of Pharmacy |
| 30910462 |
53 |
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors. |
Yanbian University |
| 31563013 |
69 |
Synthesis, anticancer activity, and molecular modeling of 1,4-naphthoquinones that inhibit MKK7 and Cdc25. |
Montana State University |
| 31541869 |
12 |
Identification of highly potent and selective Cdc25 protein phosphatases inhibitors from miniaturization click-chemistry-based combinatorial libraries. |
Shandong University |
| 31294975 |
38 |
Discovery of Novel Naphthylphenylketone and Naphthylphenylamine Derivatives as Cell Division Cycle 25B (CDC25B) Phosphatase Inhibitors: Design, Synthesis, Inhibition Mechanism, and in Vitro Efficacy against Melanoma Cell Lines. |
University of Naples Federico Ii |
| 28803043 |
10 |
Structure-based development of novel triazoles and related thiazolotriazoles as anticancer agents and Cdc25A/B phosphatase inhibitors. Synthesis, in vitro biological evaluation, molecular docking and in silico ADME-T studies. |
King Abdulaziz University |
| 28431339 |
39 |
Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells. |
Sapienza University of Rome |
| 20578711 |
19 |
Solution phase synthesis of a combinatorial library of chalcones and flavones as potent cathepsin V inhibitors. |
Universidade Federal De SaO Carlo |
| 20666436 |
56 |
Dipeptidyl-quinolone derivatives inhibit hypoxia inducible factor-1a prolyl hydroxylases-1, -2, and -3 with altered selectivity. |
Amgen |
| 16677001 |
16 |
Strategy for discovering chemical inhibitors of human cyclophilin a: focused library design, virtual screening, chemical synthesis and bioassay. |
East China Univesity of Science and Technology |
| 23306195 |
39 |
Thiolactomycin-based ß-Ketoacyl-AcpM Synthase A (KasA) Inhibitors: FRAGMENT-BASED INHIBITOR DISCOVERY USING TRANSIENT ONE-DIMENSIONAL NUCLEAR OVERHAUSER EFFECT NMR SPECTROSCOPY. |
Institute For Chemical Biology & Drug Discovery |
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