The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 23200243 |
5 |
Fluorescent ligands for adenosine receptors. |
National Institute of Diabetes and Digestive and Kidney Diseases |
| 17418915 |
48 |
QSAR study on a novel series of 8-azaadenine analogues proposed as A1 adenosine receptor antagonists. |
University of Pisa |
| 17933541 |
145 |
5'-Carbamoyl derivatives of 2'-C-methyl-purine nucleosides as selective A1 adenosine receptor agonists: affinity, efficacy, and selectivity for A1 receptor from different species. |
Universit£ |
| 15743197 |
37 |
Synthesis, biological evaluation, and molecular modeling of ribose-modified adenosine analogues as adenosine receptor agonists. |
Universit£ |
| 15214785 |
58 |
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies. |
Universit£ |
| 12383013 |
44 |
Synthesis, molecular modeling studies, and pharmacological activity of selective A(1) receptor antagonists. |
Universit£ |
| 11462973 |
47 |
3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: a new class of selective A1 adenosine receptor antagonists. |
Universit£ |
| 10956189 |
98 |
A novel class of highly potent and selective A1 adenosine antagonists: structure-affinity profile of a series of 1,8-naphthyridine derivatives. |
Universit£ |
| 9572897 |
49 |
2'-C-Methyl analogues of selective adenosine receptor agonists: synthesis and binding studies. |
Universit£ |
| 8355252 |
54 |
Adenosine A1 antagonists. 3. Structure-activity relationships on amelioration against scopolamine- or N6-((R)-phenylisopropyl)adenosine-induced cognitive disturbance. |
Kyowa Hakko Kogyo |
| 1738138 |
62 |
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential. |
Niddk |
| 1433217 |
31 |
Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists. |
National Institute of Diabetes |
| 2002461 |
37 |
1H-imidazo[4,5-c]quinolin-4-amines: novel non-xanthine adenosine antagonists. |
Center For Bio-Pharmaceutical Sciences |
| 2709373 |
63 |
Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors. |
Niddk |
| 3351850 |
46 |
125I-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors. |
University of Virginia School of Medicine |
| 2991519 |
98 |
Synthesis of xanthines as adenosine antagonists, a practical quantitative structure-activity relationship application. |
TBA |
| 6279840 |
53 |
Adenosine receptors: targets for future drugs. |
TBA |
| 21401121 |
16 |
The identification of the 2-phenylphthalazin-1(2H)-one scaffold as a new decorable core skeleton for the design of potent and selective human A3 adenosine receptor antagonists. |
Universita` Degli Studi Di Firenze |
| 20937560 |
54 |
Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligands. |
Dipartimento Di Scienze Farmaceutiche |
| | 1 |
Synthesis of 5-(3-Hydroxypropyl)-7-methoxy-2-(3‘-methoxy-4‘-hydroxyphenyl)-3- benzo[b]furancarbaldehyde, a Novel Adenosine A1 Receptor Ligand from the Root of Salvia miltiorrhiza |
TBA |
| 19301821 |
55 |
Pyrido[2,3-e]-1,2,4-triazolo[4,3-a]pyrazin-1-one as a new scaffold to develop potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies. |
Universita Di Firenze |
| 18468446 |
55 |
Synthesis, ligand-receptor modeling studies and pharmacological evaluation of novel 4-modified-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent and selective human A3 adenosine receptor antagonists. |
Universita' Di Firenze |
| 17028066 |
41 |
Synthesis, biological activity and molecular modelling of new trisubstituted 8-azaadenines with high affinity for A1 adenosine receptors. |
Università |
| 16789747 |
71 |
4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A3 adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies. |
Università |
| 16335918 |
68 |
1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives. |
Università |
| 16279775 |
61 |
Synthesis and 3D QSAR of new pyrazolo[3,4-b]pyridines: potent and selective inhibitors of A1 adenosine receptors. |
Università |
| 16099648 |
128 |
1,8-Naphthyridin-4-one derivatives as new ligands of A2A adenosine receptors. |
Dipartimento Di Scienze Farmaceutiche |
| 15163184 |
227 |
Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives. |
Università |
| 12408725 |
1 |
Synthesis and evaluation of no-carrier-added 8-cyclopentyl-3-(3-[(18)F]fluoropropyl)-1-propylxanthine ([(18)F]CPFPX): a potent and selective A(1)-adenosine receptor antagonist for in vivo imaging. |
Forschungszentrum JüLich |
| 12408713 |
54 |
Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A(1) adenosine receptor antagonists. |
Università |
| 11549462 |
11 |
Synthesis and biological data of 4-amino-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl esters, a new series of A1-adenosine receptor (A1AR) ligands. |
Facoltà |
| 10956220 |
93 |
Synthesis and structure-activity relationships of a new set of 2-arylpyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists. |
Universita' Di Firenze |
| 10737748 |
81 |
1,2,4-Triazolo[4,3-a]quinoxalin-1-one: a versatile tool for the synthesis of potent and selective adenosine receptor antagonists. |
Universita' Di Firenze |
| 9513594 |
41 |
Novel 3-aralkyl-7-(amino-substituted)-1,2,3-triazolo[4,5-d]pyrimidines with high affinity toward A1 adenosine receptors. |
Università |
| 9484505 |
12 |
A1 adenosine receptor antagonists as ligands for positron emission tomography (PET) and single-photon emission tomography (SPET). |
Forschungszentrum JüLich |
| 8071944 |
37 |
8-Azaxanthine derivatives as antagonists of adenosine receptors. |
Università |
| 6315938 |
1 |
Neurotransmitter receptor binding and drug discovery. |
TBA |
| 28789895 |
38 |
Imidazo[1,2-?]pyridines possess adenosine A |
North-West University |
| 25590533 |
245 |
Identification of a fragment-like small molecule ligand for the methyl-lysine binding protein, 53BP1. |
University of North Carolina At Chapel Hill |
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