The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26761776 |
62 |
Discovery and SAR of N-(1-((substituted piperidin-4-yl)methyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide derivatives: 5-Hydroxytryptamine receptor 4 agonist as a potent prokinetic agent. |
Sungkyunkwan University |
| 12 |
Quaternised renzapride as a potent and selective 5-HT4 receptor agonist |
TBA |
22974325 |
54 |
Identification of multiple 5-HT4 partial agonist clinical candidates for the treatment of Alzheimer's disease. |
Pfizer |
16451077 |
86 |
Pyrrolizidine esters and amides as 5-HT4 receptor agonists and antagonists. |
Pfizer |
15482914 |
25 |
Azaadamantane benzamide 5-HT4 agonists: gastrointestinal prokinetic SC-54750. |
Pfizer |
12540230 |
18 |
5-HT4 receptor ligands: applications and new prospects. |
Paris-Sud University |
10585211 |
62 |
Benzimidazole derivatives. 2. Synthesis and structure-activity relationships of new azabicyclic benzimidazole-4-carboxylic acid derivatives with affinity for serotoninergic 5-HT(3) receptors. |
Universidad Complutense |
9046352 |
86 |
New esters of 4-amino-5-chloro-2-methoxybenzoic acid as potent agonists and antagonists for 5-HT4 receptors. |
Cnrs-Biocis |
9357534 |
49 |
Novel and highly potent 5-HT3 receptor agonists based on a pyrroloquinoxaline structure. |
Universit£ |
2874226 |
27 |
Buspirone analogues. 2. Structure-activity relationships of aromatic imide derivatives. |
TBA |
| 63 |
Serotoninergic 5-HT3 and 5-HT4 receptor activities of dihydrobenzofuran carboxylic acid derivatives |
TBA |
| 26 |
Novel benzimidazole-4-carboxylic acid derivatives as potent and selective 5-HT3 receptor ligands |
TBA |
| 24 |
Synthesis and pharmacological activity of a macrocyclic benzamide |
TBA |
| 14 |
New aza(nor)adamantanes are agonists at the newly identified serotonin 5-HT4 receptor and antagonists at the 5-HT3 receptor |
TBA |
22029386 |
156 |
New serotonin 5-HT(1A) receptor agonists with neuroprotective effect against ischemic cell damage. |
Universidad Complutense De Madrid |
15801844 |
54 |
Synthesis and structure-activity relationships of a new model of arylpiperazines. 8. Computational simulation of ligand-receptor interaction of 5-HT(1A)R agonists with selectivity over alpha1-adrenoceptors. |
TBA |
| 21 |
Serotonin 5-HT4 agonist activity of a series of meso-azanoradamantane benzamides |
TBA |
| 35 |
Design of a potent 5-HT4 receptor agonist with nanomolar affinity |
TBA |
15341484 |
159 |
Synthesis and structure--activity relationship in a class of indolebutylpiperazines as dual 5-HT(1A) receptor agonists and serotonin reuptake inhibitors. |
Merck |
15149647 |
10 |
Bridgehead-methyl analog of SC-53116 as a 5-HT4 agonist. |
Pfizer |
12668005 |
21 |
Design and synthesis of S-(-)-2-[[4-(napht-1-yl)piperazin-1-yl]methyl]-1,4-dioxoperhydropyrrolo[1,2-a]pyrazine (CSP-2503) using computational simulation. A 5-HT1A receptor agonist. |
Universidad Complutense |
12383006 |
24 |
Benzimidazole derivatives. 3. 3D-QSAR/CoMFA model and computational simulation for the recognition of 5-HT(4) receptor antagonists. |
Universidad Complutense |
11597405 |
24 |
3-D-QSAR/CoMFA and recognition models of benzimidazole derivatives at the 5-HT(4) receptor. |
Universidad Complutense |
9171886 |
39 |
Arylcarbamate derivatives of 1-piperidineethanol as potent ligands for 5-HT4 receptors. |
Cnrs-Biocis |
8246239 |
84 |
Development of high-affinity 5-HT3 receptor antagonists. Structure-affinity relationships of novel 1,7-annelated indole derivatives. |
Solvay Duphar |
6581313 |
2 |
Synthesis and evaluation of a novel series of N,N-dimethylisotryptamines. |
TBA |
25965977 |
15 |
Design and synthesis of newer potential 4-(N-acetylamino)phenol derived piperazine derivatives as potential cognition enhancers. |
Panjab University |