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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
24462665 30 Discovery of novel indazole derivatives as dual angiotensin II antagonists and partial PPAR¿ agonists.EBI Glaxosmithkline
22369181 6 (Z)-2-(2-bromophenyl)-3-{[4-(1-methyl-piperazine)amino]phenyl}acrylonitrile (DG172): an orally bioavailable PPARß/d-selective ligand with inverse agonistic properties.EBI Philipps University
22133631 76 Discovery of cyclic amine-substituted benzoic acids as PPARa agonists.EBI Kyorin Pharmaceutical
21074432 25 Selective peroxisome proliferator-activated receptord isosteric selenium agonists as potent anti-atherogenic agents in vivo.EBI Seoul National University
20822906 11 A stereo-controlled synthesis of 2,4-dimethyl-4-hydroxy-16-phenylhexadecanoic acid 1,4-lactone and its PPAR activities.EBI Seoul National University
20452212 26 Glycine amides as PPARalpha agonists.EBI Bayer-Schering Pharma
19928766 425 Novel bisaryl substituted thiazoles and oxazoles as highly potent and selective peroxisome proliferator-activated receptor delta agonists.EBI The Genomics Institute of The Novartis Research Foundation
20079636 78 Synthesis and biological activities of novel indole derivatives as potent and selective PPARgamma modulators.EBI Glaxosmithkline
18947994 102 The discovery of equipotent PPARalpha/gamma dual activators.EBI Glaxosmithkline
18060776 100 Design, synthesis and evaluation of trifluoromethane sulfonamide derivatives as new potent and selective peroxisome proliferator-activated receptor alpha agonists.EBI Glaxosmithkline
17343371 27 Identification and synthesis of a novel selective partial PPARdelta agonist with full efficacy on lipid metabolism in vitro and in vivo.EBI Novo Nordisk
17157013 74 Indanylacetic acid derivatives carrying aryl-pyridyl and aryl-pyrimidinyl tail groups--new classes of PPAR gamma/delta and PPAR alpha/gamma/delta agonists.EBI Bayer Pharmaceuticals
16275077 27 Design and synthesis of substituted phenylpropanoic acid derivatives as human peroxisome proliferator-activated receptor alpha/delta dual agonists.EBI University of Tokyo
12699745 49 Novel selective small molecule agonists for peroxisome proliferator-activated receptor delta (PPARdelta)--synthesis and biological activity.EBI Glaxosmithkline
11677135 21 Identification of a series of PPAR gamma/delta dual agonists via solid-phase parallel synthesis.EBI Glaxosmithkline
11354382 42 Identification of a subtype selective human PPARalpha agonist through parallel-array synthesis.EBI Glaxosmithkline
10691680 72 The PPARs: from orphan receptors to drug discovery.EBI Glaxo Wellcome Research & Development
10508427 42 A ureido-thioisobutyric acid (GW9578) is a subtype-selective PPARalpha agonist with potent lipid-lowering activity.EBI Glaxo Wellcome Research & Development
30594433 90 Discovery of potent and selective PPAR?/? dual antagonists and initial biological studies.EBI Inception Sciences
29446942 98 Design, Synthesis, and Evaluation of a Novel Series of Indole Sulfonamide Peroxisome Proliferator Activated Receptor (PPAR)?/?/? Triple Activators: Discovery of Lanifibranor, a New Antifibrotic Clinical Candidate.EBI Inventiva