18 articles for thisTarget

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The following articles (labelled with PubMed ID or TBD) are for your review

PMID	Data	Article Title	Organization
27654218	56	Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.	Ludwig-Maximilians-Universit£T M£Nchen
25147609	18	Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor.	Hokkaido University
25698617	61	Design, synthesis and SAR studies of GABA uptake inhibitors derived from 2-substituted pyrrolidine-2-yl-acetic acids.	Ludwig-Maximilians-Universit£T M£Nchen
24112084	6	The lignan (-)-hinokinin displays modulatory effects on human monoamine and GABA transporter activities.	Drexel University College of Medicine
23886812	16	Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.	Hokkaido University
23770450	3	Synthesis of N-substituted acyclicß-amino acids and their investigation as GABA uptake inhibitors.	Zentrum F£R Pharmaforschung
21940173	32	Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.	Ludwig-Maximilians-University Munich
16246548	22	Design, synthesis, and biological evaluation of the N-diarylalkenyl-piperidinecarboxylic acid derivatives as GABA uptake inhibitors (I).	Fudan University
21353350	61	Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.	Ludwig-Maximilians-University Munich
21134748	59	Stereospecific synthesis and structure-activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors.	Glaxosmithkline
20219271	10	Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship.	Zentrum F£R Pharmaforschung
	20	On the bioactive conformation of the gaba uptake inhibitor SK&F 89976-A	TBA
30777661	42	Screening oxime libraries by means of mass spectrometry (MS) binding assays: Identification of new highly potent inhibitors to optimized inhibitors ?-aminobutyric acid transporter 1.	Ludwig-Maximilians-University M£Nchen
31117514	167	Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at ?-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters.	University of Copenhagen
30376325	50	Novel Allosteric Ligands of ?-Aminobutyric Acid Transporter 1 (GAT1) by MS Based Screening of Pseudostatic Hydrazone Libraries.	Ludwig-Maximilians-Universit£T M£Nchen
8057281	100	Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.	Synaptic Pharmaceutical
28991462	360	Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/?-Aminobutyric Acid Transporter 1 (BGT1).	University of Copenhagen