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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27654218 56 Synthesis and biological evaluation of a series of N-alkylated imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-Universit£T M£Nchen
25147609 18 Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor.EBI Hokkaido University
24112084 6 The lignan (-)-hinokinin displays modulatory effects on human monoamine and GABA transporter activities.EBI Drexel University College of Medicine
23886812 16 Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: identification of an efficient lead for potent inhibitors of GABA transports.EBI Hokkaido University
21940173 32 Aminomethyltetrazoles as potential inhibitors of the¿-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.EBI Ludwig-Maximilians-University Munich
21353350 61 Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors.EBI Ludwig-Maximilians-University Munich
21134748 59 Stereospecific synthesis and structure-activity relationships of unsymmetrical 4,4-diphenylbut-3-enyl derivatives of nipecotic acid as GAT-1 inhibitors.EBI Glaxosmithkline
20219271 10 Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship.EBI Zentrum F£R Pharmaforschung
 20 On the bioactive conformation of the gaba uptake inhibitor SK&F 89976-AEBI TBA
31117514 167 Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at ?-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters.EBI University of Copenhagen
30503411 15 Generation and screening of pseudostatic hydrazone libraries derived from 5-substituted nipecotic acid derivatives at the GABA transporter mGAT4.EBI Ludwig-Maximilians-Universit£T M£Nchen
8057281 100 Design, synthesis and evaluation of substituted triarylnipecotic acid derivatives as GABA uptake inhibitors: identification of a ligand with moderate affinity and selectivity for the cloned human GABA transporter GAT-3.EBI Synaptic Pharmaceutical
28991462 360 Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/?-Aminobutyric Acid Transporter 1 (BGT1).EBI University of Copenhagen