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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
26710088 248 Recent Progress in Histone Demethylase Inhibitors.EBI University of Oxford
26771107 113 Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 1. 3-Amino-4-pyridine Carboxylate Derivatives.EBI Glaxosmithkline
26741168 239 8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors.EBI The Institute of Cancer Research
26771203 114 Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 2. Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives.EBI Glaxosmithkline
22724510 84 Plant growth regulator daminozide is a selective inhibitor of human KDM2/7 histone demethylases.EBI University of Oxford
30343192 10 Lysine demethylase 5B (KDM5B): A potential anti-cancer drug target.EBI Zhengzhou University
27499454 22 Design and evaluation of 1,7-naphthyridones as novel KDM5 inhibitors.EBI Genentech
27476424 56 Identification of potent, selective KDM5 inhibitors.EBI Constellation Pharmaceuticals
27406798 92 Lead optimization of a pyrazolo[1,5-a]pyrimidin-7(4H)-one scaffold to identify potent, selective and orally bioavailable KDM5 inhibitors suitable for in vivo biological studies.EBI Genentech
30745098 24 Identification of novel lysine demethylase 5-selective inhibitors by inhibitor-based fragment merging strategy.EBI Kyoto Prefectural University of Medicine
31158747 257 C8-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones: Studies towards the identification of potent, cell penetrant Jumonji C domain containing histone lysine demethylase 4 subfamily (KDM4) inhibitors, compound profiling in cell-based target engagement assays.EBI Institute of Cancer Research
26682034 229 Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor.EBI University of Oxford
24325601 74 Pan-histone demethylase inhibitors simultaneously targeting Jumonji C and lysine-specific demethylases display high anticancer activities.EBI Sapienza University of Rome
28512031 65 From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors.EBI Genentech
28160945 12 In search of new a-glucosidase inhibitors: Imidazolylpyrazole derivatives.BDB University of The Punjab